Compile Data Set for Download or QSAR
maximum 50k data
Found 151 of ic50 data for polymerid = 50000354,50001081,50002497
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018100((+/-)-trans-2-hydroxy-3-(4-phenylpiperidino)-cis-d...)
Affinity DataIC50:  10nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018100((+/-)-trans-2-hydroxy-3-(4-phenylpiperidino)-cis-d...)
Affinity DataIC50:  10nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50183824(1-(2-bromobenzyl)-4-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368841(CHEMBL1204343)
Affinity DataIC50:  14nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018108(4-tert-Butyl-2-(4-phenyl-piperidin-1-yl)-cyclohexa...)
Affinity DataIC50:  20nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018094((1R,2R)-2-(4-Phenyl-piperidin-1-yl)-cyclohexanol |...)
Affinity DataIC50:  20nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368838(CHEMBL1203910)
Affinity DataIC50:  21nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368833(CHEMBL1203897)
Affinity DataIC50:  22nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368840(CHEMBL1203906)
Affinity DataIC50:  22nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368843(CHEMBL1203913)
Affinity DataIC50:  22nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368847(CHEMBL1203903)
Affinity DataIC50:  24nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368834(CHEMBL1203907)
Affinity DataIC50:  25nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50046960(1'-(4-Bromo-benzyl)-4-phenyl-[1,3']bipiperidinyl-4...)
Affinity DataIC50:  25nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50039604((+)-1''-(3-Iodo-benzyl)-4-phenyl-[1,3'']bipiperidi...)
Affinity DataIC50:  26nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368839(CHEMBL1203889)
Affinity DataIC50:  30nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368832(CHEMBL1203917)
Affinity DataIC50:  31nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368836(CHEMBL1203885)
Affinity DataIC50:  34nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368836(CHEMBL1203885)
Affinity DataIC50:  34nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50018094((1R,2R)-2-(4-Phenyl-piperidin-1-yl)-cyclohexanol |...)
Affinity DataIC50:  34nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50018078(2-(4-Phenyl-piperidin-1-yl)-cyclohexanol | 2-(4-Ph...)
Affinity DataIC50:  34nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50046947(CHEMBL172975)
Affinity DataIC50:  34nMAssay Description:Binding affinity to VAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009595(1-(4-Bromo-phenyl)-3-(4-phenyl-piperidin-1-yl)-pro...)
Affinity DataIC50:  36nMAssay Description:Displacement of [3H]vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009595(1-(4-Bromo-phenyl)-3-(4-phenyl-piperidin-1-yl)-pro...)
Affinity DataIC50:  36nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009595(1-(4-Bromo-phenyl)-3-(4-phenyl-piperidin-1-yl)-pro...)
Affinity DataIC50:  36nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368846(CHEMBL1203905)
Affinity DataIC50:  39nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018078(2-(4-Phenyl-piperidin-1-yl)-cyclohexanol | 2-(4-Ph...)
Affinity DataIC50:  40nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018078(2-(4-Phenyl-piperidin-1-yl)-cyclohexanol | 2-(4-Ph...)
Affinity DataIC50:  40nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018117(2-(4-Cyclohexyl-piperidin-1-yl)-cyclohexanol | CHE...)
Affinity DataIC50:  40nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368844(CHEMBL1203881)
Affinity DataIC50:  42nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50183823(1-(3-bromobenzyl)-3-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50:  46nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50183817(1-(2-bromobenzyl)-3-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50:  47nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018127(1-[1-(2-Hydroxy-cyclohexyl)-4-phenyl-piperidin-4-y...)
Affinity DataIC50:  50nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018134(CHEMBL20499 | N-[6-Hydroxy-7-(4-phenyl-piperidin-1...)
Affinity DataIC50:  50nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018148(3-(4-Phenyl-piperidin-1-yl)-1,2,3,4-tetrahydro-nap...)
Affinity DataIC50:  50nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018090(CHEMBL20382 | N-[6-Hydroxy-7-(4-phenyl-piperidin-1...)
Affinity DataIC50:  50nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368842(CHEMBL1203896)
Affinity DataIC50:  55nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50183813(1-benzyl-4-(4-phenylpiperazin-1-yl)piperidin-3-ol ...)
Affinity DataIC50:  57nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50183818(1-(3-bromobenzyl)-4-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50:  66nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018125(2-[4-(3-Phenyl-propyl)-piperidin-1-yl]-cyclohexano...)
Affinity DataIC50:  70nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009603(1-(3-Bromo-phenyl)-3-(4-phenyl-piperidin-1-yl)-pro...)
Affinity DataIC50:  73nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009597(1-(3-Iodo-phenyl)-3-(4-phenyl-piperidin-1-yl)-prop...)
Affinity DataIC50:  73nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50368845(CHEMBL1203911)
Affinity DataIC50:  83nMAssay Description:Inhibition of [3H]- vesamicol binding to synaptic vesicles preparation from the electric organ of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018098(5-tert-Butyl-2-(4-phenyl-piperidin-1-yl)-cyclohexa...)
Affinity DataIC50:  90nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50183812(1-(4-bromobenzyl)-3-(4-phenylpiperazin-1-yl)piperi...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50183820((E)-1-(but-2-enyl)-3-(4-phenylpiperazin-1-yl)piper...)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50183828(4-(4-phenylpiperazin-1-yl)piperidin-3-ol | CHEMBL3...)
Affinity DataIC50:  100nMAssay Description:Displacement of [3H]vesamicol from human VAChT transfected in PC12 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018080(5-(2-Oxo-hexahydro-thieno[3,4-d]imidazol-6-yl)-pen...)
Affinity DataIC50:  100nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018110(2-[4-(4-Chloro-phenyl)-piperidin-1-yl]-cyclohexano...)
Affinity DataIC50:  100nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018079(5-Amino-3-(4-phenyl-piperidin-1-yl)-1,2,3,4-tetrah...)
Affinity DataIC50:  100nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018115(2-[4-(2,5-Dimethyl-phenyl)-piperazin-1-yl]-cyclohe...)
Affinity DataIC50:  100nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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